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Found 42 from Delhi Institute of Pharmaceutical Sciences and Research
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM22985(Aralen | CHEMBL76 | CHLOROQUINE PHOSPHATE | Chloro...)
Affinity DataIC50:  20nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM22985(Aralen | CHEMBL76 | CHLOROQUINE PHOSPHATE | Chloro...)
Affinity DataIC50:  200nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Delhi Institute of Pharmaceutical Sciences and Research

LigandPNGBDBM106752(2‐[2‐(3‐fluoropyrrolidine‐...)
Affinity DataIC50:  430nMT: 2°CAssay Description:The enzyme assay was performed using DPP IV drug discovery kit (BML-AK 499; Enzo Life Sciences, Plymouth Meeting, PA, USA). The activity of test com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Delhi Institute of Pharmaceutical Sciences and Research

LigandPNGBDBM106751(2‐[2‐(3‐fluoropyrrolidine‐...)
Affinity DataIC50:  830nMT: 2°CAssay Description:The enzyme assay was performed using DPP IV drug discovery kit (BML-AK 499; Enzo Life Sciences, Plymouth Meeting, PA, USA). The activity of test com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461234(CHEMBL4226443)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461235(CHEMBL4227918)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Delhi Institute of Pharmaceutical Sciences and Research

LigandPNGBDBM106759((2S)‐2‐amino‐3‐methyl̴...)
Affinity DataIC50:  2.50E+3nMT: 2°CAssay Description:The enzyme assay was performed using DPP IV drug discovery kit (BML-AK 499; Enzo Life Sciences, Plymouth Meeting, PA, USA). The activity of test com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461235(CHEMBL4227918)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Delhi Institute of Pharmaceutical Sciences and Research

LigandPNGBDBM106753(1‐(azepan‐1‐yl)‐2‐[2...)
Affinity DataIC50:  3.47E+3nMT: 2°CAssay Description:The enzyme assay was performed using DPP IV drug discovery kit (BML-AK 499; Enzo Life Sciences, Plymouth Meeting, PA, USA). The activity of test com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461234(CHEMBL4226443)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Delhi Institute of Pharmaceutical Sciences and Research

LigandPNGBDBM106750((3-fluoropyrrolidin-1-yl) (pyrrolidin-2-yl)methano...)
Affinity DataIC50:  4.27E+3nMT: 2°CAssay Description:The enzyme assay was performed using DPP IV drug discovery kit (BML-AK 499; Enzo Life Sciences, Plymouth Meeting, PA, USA). The activity of test com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Delhi Institute of Pharmaceutical Sciences and Research

LigandPNGBDBM106756((3-Fluoro-pyrrolidin-1-yl)-[1-(2-piperidin-1-yl-et...)
Affinity DataIC50:  6.49E+3nMT: 2°CAssay Description:The enzyme assay was performed using DPP IV drug discovery kit (BML-AK 499; Enzo Life Sciences, Plymouth Meeting, PA, USA). The activity of test com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Delhi Institute of Pharmaceutical Sciences and Research

LigandPNGBDBM106754(2‐[2‐(3‐fluoropyrrolidine‐...)
Affinity DataIC50:  7.88E+3nMT: 2°CAssay Description:The enzyme assay was performed using DPP IV drug discovery kit (BML-AK 499; Enzo Life Sciences, Plymouth Meeting, PA, USA). The activity of test com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461226(CHEMBL4228534)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461226(CHEMBL4228534)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461225(CHEMBL4224867)
Affinity DataIC50:  1.43E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Delhi Institute of Pharmaceutical Sciences and Research

LigandPNGBDBM106755(2‐[2‐(3‐fluoropyrrolidine‐...)
Affinity DataIC50:  1.67E+4nMT: 2°CAssay Description:The enzyme assay was performed using DPP IV drug discovery kit (BML-AK 499; Enzo Life Sciences, Plymouth Meeting, PA, USA). The activity of test com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461237(CHEMBL4226863)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461229(CHEMBL4228490)
Affinity DataIC50:  1.86E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461239(CHEMBL4227712)
Affinity DataIC50:  1.97E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461233(CHEMBL4224976)
Affinity DataIC50:  2.09E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Delhi Institute of Pharmaceutical Sciences and Research

LigandPNGBDBM106757([1-(2-Diethylamino-ethyl)-pyrrolidin-2-yl]-(3-fluo...)
Affinity DataIC50:  2.38E+4nMT: 2°CAssay Description:The enzyme assay was performed using DPP IV drug discovery kit (BML-AK 499; Enzo Life Sciences, Plymouth Meeting, PA, USA). The activity of test com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461237(CHEMBL4226863)
Affinity DataIC50:  2.53E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461225(CHEMBL4224867)
Affinity DataIC50:  2.67E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461236(CHEMBL4228011)
Affinity DataIC50:  2.67E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461232(CHEMBL4227123)
Affinity DataIC50:  2.69E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461229(CHEMBL4228490)
Affinity DataIC50:  2.71E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461236(CHEMBL4228011)
Affinity DataIC50:  2.99E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Delhi Institute of Pharmaceutical Sciences and Research

LigandPNGBDBM106758({1-[2-(dimethylamino)ethyl]pyrrolidin-2-yl}(3- flu...)
Affinity DataIC50:  3.02E+4nMT: 2°CAssay Description:The enzyme assay was performed using DPP IV drug discovery kit (BML-AK 499; Enzo Life Sciences, Plymouth Meeting, PA, USA). The activity of test com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461239(CHEMBL4227712)
Affinity DataIC50:  3.04E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461232(CHEMBL4227123)
Affinity DataIC50:  3.38E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461230(CHEMBL4224721)
Affinity DataIC50:  3.42E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461233(CHEMBL4224976)
Affinity DataIC50:  4.16E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461230(CHEMBL4224721)
Affinity DataIC50:  4.45E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461228(CHEMBL4226325)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461231(CHEMBL4228548)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461238(CHEMBL4224700)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461238(CHEMBL4224700)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461227(CHEMBL4228230)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain-2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461228(CHEMBL4226325)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461231(CHEMBL4228548)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
Delhi Institute Of Pharmaceutical Sciences And Research

Curated by ChEMBL
LigandPNGBDBM50461227(CHEMBL4228230)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed